Preclinical Evaluation of the Pan-FGFR Inhibitor LY2874455 in FRS2-Amplified Liposarcoma

<b>Background:</b> FGFR inhibition has been proposed as treatment for dedifferentiated liposarcoma (DDLPS) with amplified <i>FRS2</i>, but we previously only demonstrated transient cytostatic effects when treating <i>FRS2</i>-amplified DDLPS cells with NVP-BGJ398....

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Bibliographic Details
Main Authors: Robert Hanes, Else Munthe, Iwona Grad, Jianhua Han, Ida Karlsen, Emmet McCormack, Leonardo A. Meza-Zepeda, Eva Wessel Stratford, Ola Myklebost
Format: Article
Language:English
Published: MDPI AG 2019-02-01
Series:Cells
Subjects:
Online Access:https://www.mdpi.com/2073-4409/8/2/189