The Different Strategies for the Radiolabeling of [<sup>211</sup>At]-Astatinated Radiopharmaceuticals

Astatine-211 (<sup>211</sup>At) has emerged as a promising radionuclide for targeted alpha therapy of cancer by virtue of its favorable nuclear properties. However, the limited in vivo stability of <sup>211</sup>At-labeled radiopharmaceuticals remains a major challenge. This...

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Bibliographic Details
Main Authors: Jie Gao, Mei Li, Jingjing Yin, Mengya Liu, Hongliang Wang, Jin Du, Jianguo Li
Format: Article
Language:English
Published: MDPI AG 2024-05-01
Series:Pharmaceutics
Subjects:
Online Access:https://www.mdpi.com/1999-4923/16/6/738