Cyclic N-locked indolicidin analogues with antimicrobial activity: Effect of ring size and fatty acid acylation

Novel antimicrobial drugs are in high demand due to the increasing emergence of multi-drug resistant bacteria. In recent years, much attention has been given to natural occurring antimicrobial peptides (AMPs) such as indolicidin (ILPWKWPWWPWRR-NH2). In this study, 19 cyclic N-locked indolicidin anal...

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Bibliographic Details
Main Authors: Abdullah Lone, Josefine Eilsø Nielsen, Peter W. Thulstrup, Reidar Lund, Paul Robert Hansen, Håvard Jenssen
Format: Article
Language:English
Published: Elsevier 2022-12-01
Series:European Journal of Medicinal Chemistry Reports
Subjects:
Online Access:http://www.sciencedirect.com/science/article/pii/S2772417422000528