Piperazine- and Piperidine-Containing Thiazolo[5,4-<i>d</i>]pyrimidine Derivatives as New Potent and Selective Adenosine A<sub>2A</sub> Receptor Inverse Agonists

The therapeutic use of A<sub>2A</sub> adenosine receptor (AR) antagonists for the treatment of neurodegenerative disorders, such as Parkinson and Alzheimer diseases, is a very promising approach. Moreover, the potential therapeutic role of A<sub>2A</sub> AR antagonists to avo...

وصف كامل

التفاصيل البيبلوغرافية
المؤلفون الرئيسيون: Flavia Varano, Daniela Catarzi, Erica Vigiani, Fabrizio Vincenzi, Silvia Pasquini, Katia Varani, Vittoria Colotta
التنسيق: مقال
اللغة:English
منشور في: MDPI AG 2020-07-01
سلاسل:Pharmaceuticals
الموضوعات:
الوصول للمادة أونلاين:https://www.mdpi.com/1424-8247/13/8/161