Enolase Inhibitors as Early Lead Therapeutics against <i>Trypanosoma brucei</i>
Glucose metabolism is critical for the African trypanosome, <i>Trypanosoma brucei</i>, serving as the lone source of ATP production for the bloodstream form (BSF) parasite in the glucose-rich environment of the host blood. Recently, phosphonate inhibitors of human enolase (ENO), the enzy...
Main Authors: | , , , , , , , , , , , , , , , , , |
---|---|
Format: | Article |
Language: | English |
Published: |
MDPI AG
2023-10-01
|
Series: | Pathogens |
Subjects: | |
Online Access: | https://www.mdpi.com/2076-0817/12/11/1290 |