Development of Androgen-Antagonistic Coumarinamides with a Unique Aromatic Folded Pharmacophore
First-generation nonsteroidal androgen receptor (AR) antagonists, such as flutamide (<b>2a</b>) and bicalutamide (<b>3</b>), are effective for most prostate cancer patients, but resistance often appears after several years due to the mutation of AR. Second-generation AR antag...
Main Authors: | , , , , , , , , |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2020-08-01
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Series: | International Journal of Molecular Sciences |
Subjects: | |
Online Access: | https://www.mdpi.com/1422-0067/21/15/5584 |