Simple and Expedient Access to Novel Fluorinated Thiazolo- and Oxazolo[3,2-<i>a</i>]pyrimidin-7-one Derivatives and Their Functionalization via Palladium-Catalyzed Reactions

Simple and Expedient Access to Novel Fluorinated Thiazolo- and Oxazolo[3,2-<i>a</i>]pyrimidin-7-one Derivatives and Their Functionalization via Palladium-Catalyzed Reactions

An efficient, versatile, and one-pot method for the preparation of novel fluorinated thiazolo- and oxazolo[3,2-<i>a</i>]pyrimidin-7-ones is described from 2-aminothiazoles or 2-amino-oxazoles and fluorinated alkynoates. This transformation, performed under transition-metal-free condition...

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Bibliographic Details
Main Authors:	Wafa Blancou, Badr Jismy, Soufiane Touil, Hassan Allouchi, Mohamed Abarbri
Format:	Article
Language:	English
Published:	MDPI AG 2022-05-01
Series:	Molecules
Subjects:	thiazolo[3,2-<i>a</i>]pyrimidin-7-ones oxazolo[3,2-<i>a</i>]pyrimidin-7-ones fluorinated alkynes regioselective one-pot reaction Suzuki-Miyaura
Online Access:	https://www.mdpi.com/1420-3049/27/9/3013

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