Rational Design, Synthesis, and Evaluation of Fluorescent CB<sub>2</sub> Receptor Ligands for Live-Cell Imaging: A Comprehensive Review
The cannabinoid receptors CB<sub>1</sub> and CB<sub>2</sub> are class A G protein-coupled receptors (GPCRs) that are activated via endogenous lipids called endocannabinoids. The endocannabinoid system (ECS) plays a critical role in the regulation of several physiological stat...
Main Authors: | , |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2023-08-01
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Series: | Pharmaceuticals |
Subjects: | |
Online Access: | https://www.mdpi.com/1424-8247/16/9/1235 |