Turning chiral peptides into a racemic supraparticle to induce the self-degradation of MDM2

Introduction: Chirality is immanent in nature, and chiral molecules can achieve their pharmacological action through chiral matching with biomolecules and molecular conformation recognition. Objectives: Clinical translation of chiral therapeutics, particularly chiral peptide molecules, has been hamp...

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Bibliographic Details
Main Authors: Wenguang Yang, Wenjia Liu, Xiang Li, Jin Yan, Wangxiao He
Format: Article
Language:English
Published: Elsevier 2023-03-01
Series:Journal of Advanced Research
Subjects:
Online Access:http://www.sciencedirect.com/science/article/pii/S2090123222001217