An Update on the Current State of SARS-CoV-2 Mac1 Inhibitors

Non-structural protein 3 (nsp3) from all coronaviruses (CoVs) contains a conserved macrodomain, known as Mac1, that has been proposed as a potential therapeutic target for CoVs due to its critical role in viral pathogenesis. Mac1 is an ADP-ribose binding protein and ADP-ribosylhydrolase that promote...

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Bibliographic Details
Main Authors: Joseph J. O’Connor, Dana Ferraris, Anthony R. Fehr
Format: Article
Language:English
Published: MDPI AG 2023-10-01
Series:Pathogens
Subjects:
Online Access:https://www.mdpi.com/2076-0817/12/10/1221