DprE1 inhibitors – a prospective target for development of antituberculosis drugs

The article reviews and analyzes 63 scientific publications devoted to new classes of antituberculosis drugs – DprE1 inhibitors. Currently, compounds BTZ-043, PBTZ-169 (makozinone), TBA-7371 and OPC-167832 are tested at different stages of clinical trials. DprE1 inhibitors are promising drugs with ant...

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Detalhes bibliográficos
Autor principal: A. V. Kukurika
Formato: Artigo
Idioma:Russian
Publicado em: New Terra Publishing House 2022-06-01
coleção:Туберкулез и болезни лёгких
Assuntos:
Acesso em linha:https://www.tibl-journal.com/jour/article/view/1644