In Silico Methods for the Discovery of Kv7.2/7.3 Channels Modulators: A Comprehensive Review

The growing interest in Kv7.2/7.3 agonists originates from the involvement of these channels in several brain hyperexcitability disorders. In particular, Kv7.2/7.3 mutants have been clearly associated with epileptic encephalopathies (DEEs) as well as with a spectrum of focal epilepsy disorders, ofte...

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Bibliographic Details
Main Authors: Claudio Stagno, Francesca Mancuso, Tania Ciaglia, Carmine Ostacolo, Anna Piperno, Nunzio Iraci, Nicola Micale
Format: Article
Language:English
Published: MDPI AG 2024-07-01
Series:Molecules
Subjects:
Online Access:https://www.mdpi.com/1420-3049/29/13/3234