Genetic function algorithm (GFA) based QSAR, molecular design, and ADMET screening to assess the antimalarial potential of Amodiaquine derivatives

The ongoing fight against endemic diseases is complicated by the increasing resistance of malaria parasites to widely used drugs. As a result, the search for more effective antimalarial treatments continues. This research focuses on developing modified Amodiaquine analogues with enhanced efficacy. A...

ver descrição completa

Detalhes bibliográficos
Principais autores: Zakari Ya’u Ibrahim, Usman Abdulfatai, Stephen Ejeh, Abduljelil Ajala, Samuel Ndaghiya Adawara, Olasupo Sabitu Babatunde
Formato: Artigo
Idioma:English
Publicado em: Elsevier 2024-12-01
coleção:The Microbe
Assuntos:
Acesso em linha:http://www.sciencedirect.com/science/article/pii/S2950194624001754