Mobocertinib: Mechanism of action, clinical, and translational science

Abstract Epidermal growth factor receptor (EGFR) exon 20 insertion (ex20ins) mutations represent ~6%–12% of all EGFR‐mutated non‐small cell lung cancer (NSCLC) cases. First‐, second‐, and third‐generation tyrosine kinase inhibitors (TKIs) have limited clinical activity against EGFR ex20ins mutations...

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Bibliographic Details
Main Authors: Michael J. Hanley, D. Ross Camidge, Robert J. Fram, Neeraj Gupta
Format: Article
Language:English
Published: Wiley 2024-03-01
Series:Clinical and Translational Science
Online Access:https://doi.org/10.1111/cts.13766