Molecular modeling study of uracil-based hydroxamic acids-containing histone deacetylase inhibitors

A quantitative structure activity relationship study was performed on a series of uracil based hydroxamide Inhibitors of maize deacetylases HD2 and histone deacetylase (Mouse HDAC1) activity for establishing quantitative relationship between biological activity and their physicochemical properties....

Full description

Bibliographic Details
Main Authors: Mukesh C. Sharma, Smita Sharma
Format: Article
Language:English
Published: Elsevier 2019-12-01
Series:Arabian Journal of Chemistry
Online Access:http://www.sciencedirect.com/science/article/pii/S1878535215000076