Modulation of the Meisenheimer complex metabolism of nitro-benzothiazinones by targeted C-6 substitution

Abstract Tuberculosis, caused by Mycobacterium tuberculosis, remains a major public health concern, demanding new antibiotics with innovative therapeutic principles due to the emergence of resistant strains. Benzothiazinones (BTZs) have been developed to address this problem. However, an unprecedent...

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Bibliographic Details
Main Authors: François Keiff, Freddy A. Bernal, Melanie Joch, Thibault J. W. Jacques dit Lapierre, Yan Li, Phil Liebing, Hans-Martin Dahse, Ivan Vilotijevic, Florian Kloss
Format: Article
Language:English
Published: Nature Portfolio 2024-07-01
Series:Communications Chemistry
Online Access:https://doi.org/10.1038/s42004-024-01235-x