Facile One-pot Protocol of Derivatization Nitropyridines: Access to 3-Acetamidopyridin-2-yl 4-methylbenzenesulfonate Derivatives

Facile One-pot Protocol of Derivatization Nitropyridines: Access to 3-Acetamidopyridin-2-yl 4-methylbenzenesulfonate Derivatives

This paper discloses an efficient one-pot protocol to convert easily accessible 3-nitropyridines to 3-acetamidopyridin-2-yl 4-methylbenzenesulfonate derivatives which are core structures of many pharmaceutical molecules. The strategy successfully combined a three-step reaction in one pot via progres...

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Bibliographic Details
Main Authors: Lin Ling, Chen Xiaoguang, Zhao Junhao, Lin Suitao, Ma Guojian, Liao Xiaojian, Feng Pengju
Format: Article
Language:English
Published: De Gruyter 2019-12-01
Series:Heterocyclic Communications
Subjects:
one-pot
[3,3]-sigmatropic rearrangement
heteroarene
pyridine derivatives
late-stage functionalization
Online Access:https://doi.org/10.1515/hc-2019-0017

Internet

https://doi.org/10.1515/hc-2019-0017

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