Rh(III)-catalyzed C–H acylmethylation of 2H-indazoles with sulfoxonium ylides

An efficient Cp*Rh(III)-catalyzed direct acylmethylation of 2H-indazoles with sulfoxonium ylides has been realized under air atmosphere via chelation-assisted strategy. This protocol enables a regioselective access to a variety of ortho-acylmethylated 2-phenylindazole derivatives in moderate to good...

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Bibliographic Details
Main Authors: Ya-Gai Wang, Jing Li, Xiao-Die Wang, Linlin Shi, Xinju Zhu, Xin-Qi Hao, Mao-Ping Song
Format: Article
Language:English
Published: Elsevier 2020-11-01
Series:Journal of Saudi Chemical Society
Subjects:
Online Access:http://www.sciencedirect.com/science/article/pii/S1319610320301174