Characterization Of Selective TRPM8 Ligands And Their Structure Activity Response (S.A.R) Relationship

PURPOSE: Transient receptor potential melastatin-8 (TRPM8) is an ion channel expressed extensively in sensory nerves, human prostate and overexpressed in a variety of cancers including prostate, breast, lung, colon and skin melanomas. It is activated by innoxious cooling and chemical stimuli. TRPM8...

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Bibliographic Details
Main Authors: Muhammad Azhar Sherkheli, Angela K. Vogt-Eisele, Daniel Bura, Leopoldo R. Beltrán Márques, Günter Gisselmann, Hanns Hatt
Format: Article
Language:English
Published: Frontiers Media S.A. 2010-07-01
Series:Journal of Pharmacy & Pharmaceutical Sciences
Online Access:https://journals.library.ualberta.ca/jpps/index.php/JPPS/article/view/7459