Synthesis and Biological Evaluation of Highly Active 7-Anilino Triazolopyrimidines as Potent Antimicrotubule Agents
Two different series of fifty-two compounds, based on 3′,4′,5′-trimethoxyaniline (<b>7a–ad</b>) and variably substituted anilines (<b>8a–v</b>) at the 7-position of the 2-substituted-[1,2,4]triazolo [1,5-<i>a</i>]pyrimidine nucleus, had moderate to potent antiprol...
Main Authors: | , , , , , , , , , , , , , |
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Format: | Article |
Language: | English |
Published: |
MDPI AG
2022-06-01
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Series: | Pharmaceutics |
Subjects: | |
Online Access: | https://www.mdpi.com/1999-4923/14/6/1191 |