Thiacalix[4]arene С-1087 is the selective inhibitor of the calcium pump of smooth muscle cells plasma membrane

Thiacalix[4]arene С-1087 is the selective inhibitor of the calcium pump of smooth muscle cells plasma membrane

The enzymatic and kinetic analyses were used to demonstrate that 5,11,17,23-tetra(trifluoro)methyl(phenylsulfonylimino)methylamino-25,27-dihexyloxy-26,28-dihydroxythiacalix[4]arene С-1087 effectively inhibited the Са2+,Mg2+-АТРase activity of the rat myometrium cells plasma membrane (І0.5 = 9.4 ± 0....

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Bibliographic Details
Main Authors: Т. О. Veklich, R. V. Rodik, О. V. Tsymbalyuk, О. V. Shkrabak, O. V. Maliuk, S. O. Karakhim, S. H. Vyshnevskyi, V. І. Kalchenko, S. O. Kosterin
Format: Article
Language:English
Published: National Academy of Sciences of Ukraine, Palladin Institute of Biochemistry 2023-12-01
Series:The Ukrainian Biochemical Journal
Subjects:
contraction-relaxation mechanokinetics
cytosolic ca(2+)
myometrium
plasma membrane са(2+)‚mg(2+)-атрase
smooth muscle cell
thiacalix[4]arene
Online Access:http://ukrbiochemjournal.org/wp-content/uploads/2023/12/Veklich_95_6.pdf

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http://ukrbiochemjournal.org/wp-content/uploads/2023/12/Veklich_95_6.pdf

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