Structural and biophysical insights into the mode of covalent binding of rationally designed potent BMX inhibitors

<p>We identified potent, functionalisable BMX inhibitors and revealed their covalent mode of binding to BMX by X-ray crystallography.</p>

Λεπτομέρειες βιβλιογραφικής εγγραφής
Κύριοι συγγραφείς:	Seixas, João D, Sousa, Bárbara B, Marques, Marta C, Guerreiro, Ana, Traquete, Rui, Rodrigues, Tiago, Albuquerque, Inês S, Sousa, Marcos FQ, Lemos, Ana R, Sousa, Pedro MF, Bandeiras, Tiago M, Wu, Di, Doyle, Shelby K, Robinson, Carol V, Koehler, Angela N, Corzana, Francisco, Matias, Pedro M, Bernardes, Gonçalo JL
Άλλοι συγγραφείς:	Koch Institute for Integrative Cancer Research at MIT
Μορφή:	Άρθρο
Γλώσσα:	English
Έκδοση:	Royal Society of Chemistry (RSC) 2022
Διαθέσιμο Online:	https://hdl.handle.net/1721.1/133096.2

Structural and biophysical insights into the mode of covalent binding of rationally designed potent BMX inhibitors ανά Seixas, João D, Sousa, Bárbara B, Marques, Marta C, Guerreiro, Ana, Traquete, Rui, Rodrigues, Tiago, Albuquerque, Inês S, Sousa, Marcos FQ, Lemos, Ana R, Sousa, Pedro MF, Bandeiras, Tiago M, Wu, Di, Doyle, Shelby K, Robinson, Carol V, Koehler, Angela N, Corzana, Francisco, Matias, Pedro M, Bernardes, Gonçalo JL

Έκδοση 2021

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