Palladium-Catalyzed Amination of Unprotected Halo-7- azaindoles

Simple and efficient procedures for the Pd-catalyzed cross-coupling of primary and secondary amines with halo-7-azaindoles(pyrrolo[2,3-b]pyridine) are presented. Previously, no general method was available to ensure the highly selective reaction of the heteroaryl halide in the presence of the unprot...

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Bibliographic Details
Main Authors: Henderson, Jaclyn L., McDermott, Sarah M., Buchwald, Stephen Leffler
Other Authors: Massachusetts Institute of Technology. Department of Chemistry
Format: Article
Language:en_US
Published: American Chemical Society (ACS) 2012
Online Access:http://hdl.handle.net/1721.1/72118
https://orcid.org/0000-0003-3875-4775