Palladium-Catalyzed N-Arylation of 2-Aminothiazoles

A method for the Pd-catalyzed coupling of 2-aminothiazole derivatives with aryl bromides and triflates is described. Significantly, for this class of nucleophiles, the coupling exhibits a broad substrate scope and proceeds with a reasonable catalyst loading. Furthermore, an interesting effect of ace...

詳細記述

書誌詳細
主要な著者: McGowan, Meredeth A., Henderson, Jaclyn L., Buchwald, Stephen Leffler
その他の著者: Massachusetts Institute of Technology. Department of Chemistry
フォーマット: 論文
言語:en_US
出版事項: American Chemical Society (ACS) 2013
オンライン・アクセス:http://hdl.handle.net/1721.1/81945
https://orcid.org/0000-0003-3875-4775