Synthesis of Spirocyclic Indolines by Interruption of the Bischler–Napieralski Reaction
The development of a versatile method for the synthesis of spirocyclic pyrrolidinoindolines is discussed. Treatment of N-acyltryptamines with trifluoromethanesulfonic anhydride–2-chloropyridine reagent combination affords highly persistent spiroindoleninium ions that are subject to intra- and interm...
Main Authors: | Medley, Jonathan William, Movassaghi, Mohammad |
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Other Authors: | Massachusetts Institute of Technology. Department of Chemistry |
Format: | Article |
Language: | en_US |
Published: |
American Chemical Society (ACS)
2015
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Online Access: | http://hdl.handle.net/1721.1/95519 https://orcid.org/0000-0003-3080-1063 |
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