Recent progress in histone demethylase inhibitors

There is increasing interest in targeting histone N-methyl-lysine demethylases (KDMs) with small molecules both for the generation of probes for target exploration and for therapeutic purposes. Here we update on previous reviews on the inhibition of the lysine-specific demethylases (LSDs or KDM1s) a...

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Bibliographic Details
Main Authors: McAllister, T, England, KS, Hopkinson, R, Brennan, PE, Kawamura, A, Schofield, CJ
Format: Journal article
Language:English
Published: American Chemical Society 2016