Dimerization of lithiated terminal aziridines.
Let's get together: Dimerization of enantiopure terminal aziridines by lithiation gives efficiently N-protected 2-ene-1,4-diamines with complete selectivity for the E olefin (see scheme). The usefulness of the method was demonstrated in a concise synthesis of (R,S,S,R)-2,5-diamino-1,6-diphenylh...
Main Authors: | , |
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Format: | Journal article |
Language: | English |
Published: |
2006
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