Palladium-catalyzed allylic fluorination.
Mild and rapid: The title reaction is presented and its applicability to 18F radiolabeling is demonstrated (see scheme; TBAF=tetra-n- butylammonium fluoride, THF=tetrahydrofuran, dba=dibenzylideneacetone). The use of p-nitrobenzoate as the leaving group is significant to the success of this catalyti...
Main Authors: | , , , , , , , , |
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Format: | Journal article |
Language: | English |
Published: |
2011
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