Metal free fluoroamination of allylsilanes: A route to 3-fluoropyrrolidines
The intramolecular fluoroamination of homoallylic amines activated by a triisopropylsilyl or p-tolyldiisopropylsilyl group was successfully performed in the presence of Selectfluor® in acetonitrile leading to anti or syn 3-fluoropyrrolidines. The stereochemical outcome of these fluorocyclizations is...
Main Authors: | , , |
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Format: | Journal article |
Language: | English |
Published: |
2012
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