A stereoselective oxy-Michael route to protected beta-aryl-beta-hydroxy-alpha-amino acids
The stereoselective oxy-Michael addition of the 'naked' anion of (5)-6-methyl tetrahydropyran-2-ol to α-nitro-α,β-unsaturated esters followed by reduction and in situ protection of the corresponding amine provides a new and efficient route to protected β-aryl-β-hydroxy- α-amino acids. © Ge...
| Hoofdauteurs: | , , |
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| Formaat: | Journal article |
| Taal: | English |
| Gepubliceerd in: |
2006
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