Structure-activity studies of a macrocyclic peptide inhibitor of histone lysine demethylase 4A
The combination of genetic code reprogramming and mRNA display is a powerful approach for the identification of macrocyclic peptides with high affinities to a target of interest. We have previously used such an approach to identify a potent inhibitor (CP2) of the human KDM4A and KDM4C lysine demethy...
Huvudupphovsmän: | , , , , |
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Materialtyp: | Journal article |
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Elsevier
2018
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