Design, synthesis and structure-activity relationships of 3,5-diaryl-1H-pyrazoles as inhibitors of arylamine N-acetyltransferase.
The synthesis and inhibitory potencies of a novel series of 3,5-diaryl-1H-pyrazoles as specific inhibitors of prokaryotic arylamine N-acetyltransferase enzymes is described. The series is based on hit compound 1 3,5-diaryl-1H-pyrazole identified from a high-throughout screen that has been carried ou...
وصف كامل
التفاصيل البيبلوغرافية
| المؤلفون الرئيسيون: |
Fullam, E,
Talbot, J,
Abuhammed, A,
Westwood, I,
Davies, S,
Russell, A,
Sim, E |
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| التنسيق: | Journal article
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| اللغة: | English |
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| منشور في: |
2013
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