Orthogonal N,N-deprotection strategies of beta-amino esters
β-Amino esters derived from the stereoselective conjugate addition of homochiral lithium N-benzyl-N-α-methyl-4-methoxybenzylamide to α,β-unsaturated esters may be orthogonally mono-N-deprotected under either oxidative or acid-promoted reaction conditions. Further oxidative deprotection affordsβ-amin...
Main Authors: | , , , , |
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Format: | Journal article |
Language: | English |
Published: |
2001
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