Orthogonal N,N-deprotection strategies of beta-amino esters
β-Amino esters derived from the stereoselective conjugate addition of homochiral lithium N-benzyl-N-α-methyl-4-methoxybenzylamide to α,β-unsaturated esters may be orthogonally mono-N-deprotected under either oxidative or acid-promoted reaction conditions. Further oxidative deprotection affordsβ-amin...
Main Authors: | Bull, S, Davies, S, Kelly, P, Gianotti, M, Smith, A |
---|---|
Format: | Journal article |
Language: | English |
Published: |
2001
|
Similar Items
-
Selective deprotection strategies to N-(alpha-methylbenzyl)-beta-amino esters and derived beta lactams
by: Davies, S, et al.
Published: (1998) -
Asymmetric synthesis of beta-haloaryl beta-amino acid derivatives
by: Bull, S, et al.
Published: (2001) -
Asymmetric synthesis of beta-pyridyl-beta-amino acid derivatives
by: Bull, S, et al.
Published: (2002) -
Trading N and O: asymmetric syntheses of beta-hydroxy-alpha-amino acids via alpha-hydroxy-beta-amino esters
by: Davies, S, et al.
Published: (2013) -
Observations on the deprotection of pinanediol and pinacol boronate esters via fluorinated intermediates.
by: Inglis, SR, et al.
Published: (2010)