Pyrrolidinones derived from (S)-pyroglutamic acid. Part 2. Conformationally constrained kainoid analogues

Pyrrolidinones derived from (S)-pyroglutamic acid. Part 2. Conformationally constrained kainoid analogues

Novel conformationally constrained glutamate analogues are readily available from (S)-pyroglutamic acid using a bicyclic lactam as a synthetic template; diastereocontrolled modification of the pyrrolidine ring using a sequential conjugate addition-substitution strategy permits access to several kain...

पूर्ण विवरण

ग्रंथसूची विवरण
मुख्य लेखकों:	Dyer, J, King, A, Keeling, S, Moloney, M
स्वरूप:	Journal article
भाषा:	English
प्रकाशित:	2000

समान संसाधन

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Direct versatile route to conformationally constrained glutamate analogues
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ENANTIOSELECTIVE KAINOID SYNTHESIS BY COBALT-MEDIATED CYCLIZATION OF AN AMINO-ACID DERIVATIVE
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Molecular Dynamics Simulation Reveal the Structure–Activity Relationships of Kainoid Synthases
द्वारा: Zeyu Fan, और अन्य
प्रकाशित: (2024-07-01)

Metabolic Acidosis Due To Pyroglutamic Acid
द्वारा: Maria João Raposo Linhares Serpa, और अन्य
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