5,5-Fused thiophene gamma-lactams as templates for serine protease inhibition.
Novel 5,5-fused thiophene lactams are potent inhibitors and acylating agents of HNE and PPE.
Главные авторы: | Migaud, M, Wilmouth, R, Mills, G, Wayne, G, Risley, C, Chambers, C, Macdonald, S, Schofield, C |
---|---|
Формат: | Journal article |
Язык: | English |
Опубликовано: |
2002
|
Схожие документы
-
5,5-Fused thiophene gamma-lactams as templates for serine protease inhibition.
по: Migaud, M, и др.
Опубликовано: (2002) -
Mechanistic insights into the inhibition of serine proteases by monocyclic lactams.
по: Wilmouth, R, и др.
Опубликовано: (1999) -
Structural analyses on intermediates in serine protease catalysis.
по: Liu, B, и др.
Опубликовано: (2006) -
Thiophene-fused γ-lactams inhibit the SARS-CoV-2 main protease via reversible covalent acylation
по: Gayatri, и др.
Опубликовано: (2024) -
beta-Sultams - A novel class of serine protease inhibitors
по: Beardsell, M, и др.
Опубликовано: (2001)