In vitro activities of 2,4-diaminoquinazoline and 2,4-diaminopteridine derivatives against Plasmodium falciparum

The activities of 28 6-substituted 2,4-diaminoquinazolines, 2,4-diamino-5,6,7,8-tetrahydroquinazolines, and 2,4-diaminopteridines against Plasmodium falciparum were tested. The 50% inhibitory concentrations (IC 50s) of six compounds were <50 nM, and the most potent compound was 2,4-diamino-5-...

Полное описание

Библиографические подробности
Главные авторы: Ommeh, S, Nduati, E, Mberu, E, Kokwaro, G, Marsh, K, Rosowsky, A, Nzila, A
Формат: Journal article
Язык:English
Опубликовано: 2004