SULFATION PATHWAYS: Steroid sulphatase inhibition via aryl sulphamates: clinical progress, mechanism and future prospects

SULFATION PATHWAYS: Steroid sulphatase inhibition via aryl sulphamates: clinical progress, mechanism and future prospects

Steroid sulphatase is an emerging drug target for the endocrine therapy of hormone-dependent diseases, catalysing oestrogen sulphate hydrolysis to oestrogen. Drug discovery, developing the core aryl O-sulphamate pharmacophore, has led to steroidal and non-steroidal drugs entering numerous clinical t...

Бүрэн тодорхойлолт

Номзүйн дэлгэрэнгүй
Үндсэн зохиолч:	Potter, B
Формат:	Journal article
Хэл сонгох:	English
Хэвлэсэн:	BioScientifica 2018

Ижил төстэй зүйлс

SULFATION PATHWAYS: Steroid sulfatase inhibition by aryl sulfamates: clinical progress, mechanism and future prospects
-н: Potter, B
Хэвлэсэн: (2018)

Steroid Sulphatase and Its Inhibitors: Past, Present, and Future
-н: Paul A. Foster
Хэвлэсэн: (2021-05-01)

New potent steroid sulphatase inhibitors based on 6-(1-phenyl-1H-1,2,3-triazol-4-yl)naphthalen-2-yl sulphamate derivatives
-н: Olga Ciupak, зэрэг
Хэвлэсэн: (2021-01-01)

Placental steroid sulphatase deficiency: an approach to antenatal care and delivery
-н: Frieda-Elsje Dreyer, зэрэг
Хэвлэсэн: (2018-11-01)

Recent progress in the development of steroid sulphatase inhibitors – examples of the novel and most promising compounds from the last decade
-н: Mateusz Daśko, зэрэг
Хэвлэсэн: (2020-01-01)

Identification of oestrone sulphatase inhibitors in breast cyst fluid
-н: Lai, Leslie Charles, зэрэг
Хэвлэсэн: (2002)

Effect of NaCl on the properties of sulphamic acid single crystals
-н: J. Arumugam, зэрэг
Хэвлэсэн: (2019-07-01)

Investigations on Growth, Optical and Thermal Properties of Sulphamic Acid Single Crystals
-н: D. Jaishree, зэрэг
Хэвлэсэн: (2014-01-01)

Effect of Breast Cyst Fluid on Oestrone Sulphatase Activity in Breast Cancer Celllines
-н: El-Sadig, Rasha El-Hag
Хэвлэсэн: (2000)

Effect of Aquo-glycolic Media and Added Anions on the Anodization of Zircaloy-4 in Sulphamic Acid
-н: Viplav Duth Shukla, зэрэг
Хэвлэсэн: (2011-01-01)

Identification of oestrone sulphatase inhibitors in breast cyst fluid: a new treatment for breast cancer
-н: Lai, L. C.
Хэвлэсэн: (1999)

Growth, characterization, and anti-bacterial activity of l-methionine supplemented with sulphamic acid single crystals
-н: Vithel Friedelin R. S., зэрэг
Хэвлэсэн: (2024-02-01)

Insights into the binding mode of sulphamates and sulphamides to hCA II: crystallographic studies and binding free energy calculations
-н: Giuseppina De Simone, зэрэг
Хэвлэсэн: (2017-01-01)

Radioiodination of Aryl-Alkyl Cyclic Sulfates
-н: Mikhail I. Papisov, зэрэг
Хэвлэсэн: (2012-11-01)

2-Methoxyestradiol-bis-sulphamate refrains from inducing apoptosis and autophagy in a non-tumorigenic breast cell line
-н: Visagie Michelle H, зэрэг
Хэвлэсэн: (2012-08-01)

Microwave-assisted solvent-free one pot synthesis of isobenzofuran-1(3H)-ones using sulphamic acid catalyst
-н: Samruddhi S. Zambre, зэрэг
Хэвлэсэн: (2016-11-01)

Steroid Sulfation in Neurodegenerative Diseases
-н: Jana Vitku, зэрэг
Хэвлэсэн: (2022-02-01)

<it>In vitro </it>effects of 2-methoxyestradiol-bis-sulphamate on reactive oxygen species and possible apoptosis induction in a breast adenocarcinoma cell line
-н: Visagie Michelle H, зэрэг
Хэвлэсэн: (2011-12-01)

Aryl Hydrocarbon Receptor Inhibition Restores Indoxyl Sulfate-Mediated Endothelial Dysfunction in Rat Aortic Rings
-н: Cindy Nguyen, зэрэг
Хэвлэсэн: (2022-01-01)

Steroid Sulfatase Inhibition: From Concept to Clinic and Beyond
-н: Barry V L Potter
Хэвлэсэн: (2019-08-01)

Sulfated and Sulfur-Containing Steroids and Their Pharmacological Profile
-н: Tatyana A. Pounina, зэрэг
Хэвлэсэн: (2021-04-01)

Multiplexing Iduronate-2-Sulphatase (MPS-II) into a 7-Plex Lysosomal Storage Disorder MS/MS Assay Using Cold-Induced Phase Separation
-н: Elya Courtney, зэрэг
Хэвлэсэн: (2023-06-01)

Inhibition of Human Osteoclast Differentiation by Kynurenine through the Aryl-Hydrocarbon Receptor Pathway
-н: So-Yeon Kim, зэрэг
Хэвлэсэн: (2021-12-01)

MECHANISMS OF OSTEOBLAST INHIBITION BY STEROIDS
-н: Hulley, P
Хэвлэсэн: (2004)

Assembly of (hetero)aryl sulfilimines via copper-catalyzed enantioselective S-arylation of sulfenamides with (hetero)aryl Iodides
-н: Mingchuang He, зэрэг
Хэвлэсэн: (2025-03-01)

Role of Chondroitin Sulfate Proteoglycan 5 in Steroid-Induced Cataract
-н: Woong-Sun Yoo, зэрэг
Хэвлэсэн: (2023-06-01)

Pregnenolone Sulfate: From Steroid Metabolite to TRP Channel Ligand
-н: Christian Harteneck
Хэвлэсэн: (2013-09-01)

Dual processing of sulfated steroids in the olfactory system of an anuran amphibian
-н: Alfredo eSansone, зэрэг
Хэвлэсэн: (2015-09-01)

Generation of Aryl Radicals from Aryl Hydrazines via Catalytic Iodine in Air: Arylation of Substituted 1,4-Naphthoquinones
-н: Saibal Sar, зэрэг
Хэвлэсэн: (2020-02-01)

Empowering nanophotonic applications via artificial intelligence: pathways, progress, and prospects
-н: Chen Wei, зэрэг
Хэвлэсэн: (2025-02-01)

Synthesis of 2-aryl-benzothiazoles via Ni-catalyzed coupling of benzothiazoles and aryl sulfamates
-н: Yu Xiaofeng, зэрэг
Хэвлэсэн: (2020-02-01)

Dehydroepiandrosterone sulfate (DHEAS) stimulates the first step in the biosynthesis of steroid hormones.
-н: Jens Neunzig, зэрэг
Хэвлэсэн: (2014-01-01)

Higher steroid sulfation is linked to successful weight loss in obese children
-н: Thomas Reinehr, зэрэг
Хэвлэсэн: (2018-10-01)

High levels of oxysterol sulfates in serum of patients with steroid sulfatase deficiency[S]
-н: Alberto Sánchez-Guijo, зэрэг
Хэвлэсэн: (2015-02-01)

Rutaecarpine Inhibits U87 Glioblastoma Cell Migration by Activating the Aryl Hydrocarbon Receptor Signaling Pathway
-н: Yiyun Liu, зэрэг
Хэвлэсэн: (2021-12-01)

Integrated catalysis opens new arylation pathways via regiodivergent enzymatic C–H activation
-н: Jonathan Latham, зэрэг
Хэвлэсэн: (2016-06-01)

Isoalantolactone suppresses gallbladder cancer progression via inhibiting the ERK signalling pathway
-н: Xingyu Lv, зэрэг
Хэвлэсэн: (2023-12-01)

Chrysophanol Inhibits the Progression of Diabetic Nephropathy via Inactivation of TGF-β Pathway
-н: Guo C, зэрэг
Хэвлэсэн: (2020-11-01)

Aryl Hydrocarbon Receptor: From Homeostasis to Tumor Progression
-н: Claudia Rejano-Gordillo, зэрэг
Хэвлэсэн: (2022-04-01)

1-Methyl-D-tryptophan activates aryl hydrocarbon receptor, a pathway associated with bladder cancer progression
-н: Luiz Henrique Gomes Matheus, зэрэг
Хэвлэсэн: (2020-09-01)