Access to the bicyclic core of isatisine, and an investigation of its antibacterial activity
A chemoselective Dieckmann ring closure using an oxazolidine derived from serine may be used to generate a tetramic acid, the further manipulation of which by reduction and ring closure leads to the bicyclic core of isatisine; depending on the nature of the ring closing electrophile, different diast...
Main Authors: | , , , , |
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Format: | Journal article |
Language: | English |
Published: |
2011
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