RVX-208, an inhibitor of BET transcriptional regulators with selectivity for the second bromodomain
Bromodomains have emerged as attractive candidates for the development of inhibitors targeting gene transcription. Inhibitors of the bromo and extraterminal (BET) family recently showed promising activity in diverse disease models. However, the pleiotropic nature of BET proteins regulating tissue-sp...
| Main Authors: | , , , , , , , , , , , , , , |
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| Format: | Journal article |
| Published: |
2013
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