Synthesis and biological evaluation of phospholane and dihydrophosphole analogues of the glutamate receptor agonist AP4

The syntheses and preliminary pharmacological characterisation of two novel cyclic phosphinic acid-containing amino acids designed as conformationally restricted analogues of the metabotropic glutamate receptor agonist AP4 (1) are reported.

Библиографические подробности
Главные авторы:	Conway, S, Miller, J, Bond, A, Clark, B, Jane, D
Формат:	Journal article
Язык:	English
Опубликовано:	2002

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