The role of BET attenuation in melanoma
Bromodomain and extra-terminal (BETs) proteins function as epigenetic readers by docking onto acetylated lysine residues (Kac) on histone tails via tandem bromodomains (BRDs), and recruiting protein binding partners via an extra-terminal recruitment domain (ET). Targeting BET BRDs is efficacious in...
Váldodahkki: | |
---|---|
Eará dahkkit: | |
Materiálatiipa: | Oahppočájánas |
Giella: | English |
Almmustuhtton: |
2020
|
Fáttát: |