Synthesis and evaluation of delta-lactams (piperazones) as elastase inhibitors.

A series of monocyclic delta-lactams (piperazones) was prepared and analysed as inhibitors of porcine pancreatic elastase and human neutrophil elastase.

Bibliographic Details
Main Authors: Seibel, J, Brown, D, Amour, A, Macdonald, S, Oldham, N, Schofield, C
Format: Journal article
Language:English
Published: 2003