Specific CLK inhibitors from a novel chemotype for regulation of alternative splicing.

Specific CLK inhibitors from a novel chemotype for regulation of alternative splicing.

عرض إصدارات أخرى (1)

There is a growing recognition of the importance of protein kinases in the control of alternative splicing. To define the underlying regulatory mechanisms, highly selective inhibitors are needed. Here, we report the discovery and characterization of the dichloroindolyl enaminonitrile KH-CB19, a pote...

وصف كامل

التفاصيل البيبلوغرافية
المؤلفون الرئيسيون:	Fedorov, O, Huber, K, Eisenreich, A, Filippakopoulos, P, King, O, Bullock, A, Szklarczyk, D, Jensen, L, Fabbro, D, Trappe, J, Rauch, U, Bracher, F, Knapp, S
التنسيق:	Journal article
اللغة:	English
منشور في:	2011

مواد مشابهة

Specific CLK inhibitors from a novel chemotype for regulation of alternative splicing.
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منشور في: (2011)

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Kinase domain insertions define distinct roles of CLK kinases in SR protein phosphorylation
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