An approach to the generation of simple analogues of the antitumour agent spicamycin.
The one-step glycosylation of arylamines in acidic medium is extended to adenine derivatives for the first time, providing a considerable improvement over existing reactions. This method is used to prepare some rhamnospicamycin analogues containing different base moieties. Results suggest that this...
Main Authors: | , |
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Format: | Journal article |
Language: | English |
Published: |
2003
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