The pharmacological properties of the imidazobenzodiazepine, FG 8205, a novel partial agonist at the benzodiazepine receptor.

1. The pharmacological properties of the benzodiazepine receptor ligand, FG 8205 (7-chloro-5,6-dihydro-5-methyl-6-oxo-3-(5-isopropyl-1,2,4-oxadiazol++ +-3-yl)-4H- imidazol[1,5a][1,4]benzodiazepine) have been examined. 2. FG 8205 potently displaced [3H]-flumazenil binding in rat cortical membranes wi...

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Bibliographic Details
Main Authors: Tricklebank, MD, Honoré, T, Iversen, S, Kemp, J, Knight, A, Marshall, G, Rupniak, N, Singh, L, Tye, S, Watjen, F
Format: Journal article
Language:English
Published: 1990