Tandem copper-catalysed aryl and alkenyl amination reactions: the synthesis of N-functionalised indoles.
A Cu-diamine complex effectively catalyses tandem C-N bond formation on 2-(2-haloalkenyl)-aryl halide substrates, to deliver a series of N-functionalised indoles. Anilines, amides and carbamates are all effective coupling partners under the developed conditions.
Prif Awduron: | Hodgkinson, R, Schulz, J, Willis, M |
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Fformat: | Journal article |
Iaith: | English |
Cyhoeddwyd: |
2009
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Eitemau Tebyg
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