Twofold radical-based synthesis of N,C-difunctionalized bicyclo[1.1.1]pentanes
<p>Bicyclo[1.1.1]pentylamines (BCPAs) are of growing importance to the pharmaceutical industry as sp<sup>3</sup>-rich bioisosteres of anilines and <em>N</em>-<em>tert</em>-butyl groups. Here we report a facile synthesis of 1,3-disubstituted BCPAs us...
| Main Authors: | , , , , , |
|---|---|
| Format: | Journal article |
| Language: | English |
| Published: |
American Chemical Society
2021
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