Intramolecular cyclopropanation of unsaturated terminal aziridines.
Regio- and stereoselective deprotonation of bishomoallylic terminal N-Bus (Bus=tert-butylsulfonyl)-protected aziridines generate aziridinyl anions that undergo diastereoselective intramolecular cyclopropanation giving trans-2-aminobicyclo[3.1.0]hexanes in good to excellent yields.
| Main Authors: | , , |
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| Format: | Journal article |
| Language: | English |
| Published: |
2006
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