Hoe 140 and pseudo-irreversible antagonism in the rat vas deferens in vitro.

The effects of bradykinin and the bradykinin B(2) receptor antagonists D-Arg-[Hyp(3),Thi(5,8),D-Phe(7)]-bradykinin (NPC 349) and D-Arg-[Hyp(3),Thi(5),D-Tic(7),Oic(8)]-bradykinin (Hoe 140) were examined in the electrically-stimulated rat vas deferens. Cumulative additions of bradykinin (1-3000 nM) pr...

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Bibliographic Details
Main Authors: Asghar, A, Wheeldon, A, Coleman, R, Bountra, C, McQueen, D
Format: Journal article
Language:English
Published: 2000